Thursday 16 July 2009

Flaxel




Flaxel may be available in the countries listed below.


Ingredient matches for Flaxel



Celecoxib

Celecoxib is reported as an ingredient of Flaxel in the following countries:


  • Peru

International Drug Name Search

Wednesday 15 July 2009

Lexiscan


Lexiscan is a brand name of regadenoson, approved by the FDA in the following formulation(s):


LEXISCAN (regadenoson - solution; intravenous)



  • Manufacturer: ASTELLAS

    Approval date: April 10, 2008

    Strength(s): 0.4MG/5ML (0.08MG/ML) [RLD]

Has a generic version of Lexiscan been approved?


No. There is currently no therapeutically equivalent version of Lexiscan available.


Note: Fraudulent online pharmacies may attempt to sell an illegal generic version of Lexiscan. These medications may be counterfeit and potentially unsafe. If you purchase medications online, be sure you are buying from a reputable and valid online pharmacy. Ask your health care provider for advice if you are unsure about the online purchase of any medication.

See also: About generic drugs.




Related Patents


Patents are granted by the U.S. Patent and Trademark Office at any time during a drug's development and may include a wide range of claims.




  • N-pyrazole A2A adenosine receptor agonists
    Patent 6,403,567
    Issued: June 11, 2002
    Inventor(s): Jeff A.; Zablocki & Elfatih O.; Elzein & Venkata P.; Palle
    Assignee(s): CV Therapeutics, Inc.
    2-adenosine N-pyrazole compositions having the following formula: and methods for using the compositions as A2A receptor agonists to stimulate mammalian coronary vasodilatation for therapeutic purposes and for purposes of imaging the heart.
    Patent expiration dates:

    • April 10, 2022
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART
      ✓ 
      Drug substance
      ✓ 
      Drug product




  • 2-(N-pyrazolo)adenosines with application as adenosine A2A receptor agonists
    Patent 6,642,210
    Issued: November 4, 2003
    Inventor(s): Jeff A.; Zablocki & Elfatih O.; Elzein & Venkata P.; Palle
    Assignee(s): CV Therapeutics, Inc.
    N-pyrazole substituted 2-adenosine compounds and methods for using the compounds as A2A-adenosine receptor agonists useful to stimulate mammalian coronary vasodilation for therapeutic purposes and as adjuncts in cardiological imaging.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART
      ✓ 
      Drug substance
      ✓ 
      Drug product




  • N-pyrazole A2A receptor agonists
    Patent 7,144,872
    Issued: December 5, 2006
    Inventor(s): Zablocki; Jeff A. & Elzein; Elfatih O. & Palle; Venkata & Belardinelli; Luiz
    Assignee(s): CV Therapeutics, Inc.
    This specification discloses 2-adenosine N-pyrazole compounds having the following formula: and methods for using the compounds as A2A receptor agonists to stimulate mammalian coronary vasodilatation for therapeutic purposes and for purposes of imaging the heart.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD OF PRODUCING CORONARY VASODILATION WITHOUT PERIPHERAL VASODILATION
      ✓ 
      Drug substance
      ✓ 
      Drug product


    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART
      ✓ 
      Drug substance
      ✓ 
      Drug product


    • June 22, 2019
      ✓ 
      Patent use: METHOD OF MYOCARDIAL IMAGING
      ✓ 
      Drug substance
      ✓ 
      Drug product




  • N-pyrazole A2A receptor agonists
    Patent 7,183,264
    Issued: February 27, 2007
    Inventor(s): Zablocki; Jeff & Elzein; Elfatih O. & Palle; Venkata P. & Belardinelli; Luiz
    Assignee(s): CV Therapeutics, Inc.
    2-adenosine N-pyrazole compounds having the following formula: and methods for using the compounds as A2A receptor agonists to stimulate mammalian coronary vasodilatation for therapeutic purposes and for purposes of imaging the heart are disclosed.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD OF PRODUCING CORONARY VASODILATION WITHOUT PERIPHERAL VASODILATION
      ✓ 
      Drug product


    • June 22, 2019
      ✓ 
      Patent use: METHOD OF MYOCARDIAL IMAGING
      ✓ 
      Drug product


    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART
      ✓ 
      Drug product




  • Myocardial perfusion imaging method
    Patent 7,582,617
    Issued: September 1, 2009
    Inventor(s): Belardinelli; Luiz & Blackburn; Brent K. & Gao; Zhenhai
    Assignee(s): CV Therapeutics, Inc.
    The present invention provides a method for using the partial adenosine A2A receptor agonists having the following structure in myocardiological perfusion imaging.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: A METHOD OF MYOCARDIAL PERFUSION IMAGING AND INCREASING CORONARY BLOOD FLOW




  • Use of A2A adenosine receptor agonists
    Patent 7,655,636
    Issued: February 2, 2010
    Inventor(s): Gordi; Toufigh & Olmsted; Ann Walls & Lieu; Hsiao Dee & Belardinelli; Luiz
    Assignee(s): Gilead Palo Alto, Inc.
    The present invention relates to methods for producing coronary vasodilation with little peripheral vasodilation by administering doses of a pharmaceutical composition including regadenoson, named (1-{9-[(4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-6-aminopurin-2-yl}pyrazol-4-yl)-N-methylcarboxamide, — an adenosine A2A receptor agonist — to a human in an amount sufficient to increase the average coronary peak flow velocity by at least about 16.5 cm/sec.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART




  • N-pyrazole A2A receptor agonists
    Patent 7,655,637
    Issued: February 2, 2010
    Inventor(s): Zablocki; Jeff A. & Elzein; Elfatih O. & Palle; Venkata & Belardinelli; Luiz
    Assignee(s): Gilead Palo Alto, Inc.
    2-adenosine N-pyrazole compounds having the following formula: wherein R1═CH2OH; R2 is hydrogen; R3 is selected from the group consisting of CO2R20; —CONR7R8 ,and aryl wherein the aryl substituent is optionally substituted with one substituent selected from the group consisting of halo, C 1-3alkyl and OR20;R4 is hydrogen; R7 is selected from hydrogen, and C1-3alkyl; R8 is hydrogen; and R20 is selected from hydrogen and methyl as well as methods for using the compositions as A2A receptor agonists to stimulate mammalian coronary vasodilatation for therapeutic purposes and for purposes of imaging the heart are disclosed.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONOARY VASODILATION FOR PURPOSES OF IMAGING THE HEART
      ✓ 
      Drug substance
      ✓ 
      Drug product




  • Myocardial perfusion imaging method
    Patent 7,683,037
    Issued: March 23, 2010
    Inventor(s): Belardinelli; Luiz
    Assignee(s): Gilead Palo Alto, Inc.
    The present invention relates to methods for myocardial imaging by administering at least one 2-adenosine N-pyrazole, 2-adenosine C-pyrazole or a combination thereof A2A adenosine receptor agonist to a human undergoing myocardial imaging. The invention also relates to methods of producing coronary vasodilation without significant peripheral vasodilation by administering at least one 2-adenosine N-pyrazole, 2-adenosine C-pyrazole or a combination thereof adenosine A2A adenosine receptor agonist to a human.
    Patent expiration dates:

    • June 22, 2019
      ✓ 
      Patent use: METHOD FOR STIMULATING CORONARY VASODILATION FOR PURPOSES OF IMAGING THE HEART



Related Exclusivities

Exclusivity is exclusive marketing rights granted by the FDA upon approval of a drug and can run concurrently with a patent or not. Exclusivity is a statutory provision and is granted to an NDA applicant if statutory requirements are met.

  • Exclusivity expiration dates:
    • April 10, 2013 - NEW CHEMICAL ENTITY

See also...

  • Lexiscan Consumer Information (Drugs.com)
  • Lexiscan Consumer Information (Cerner Multum)
  • Lexiscan Advanced Consumer Information (Micromedex)
  • Regadenoson Consumer Information (Cerner Multum)
  • Regadenoson Intravenous Advanced Consumer Information (Micromedex)

Tuesday 14 July 2009

Exlutena




Exlutena may be available in the countries listed below.


Ingredient matches for Exlutena



Lynestrenol

Lynestrenol is reported as an ingredient of Exlutena in the following countries:


  • Sweden

International Drug Name Search

Monday 6 July 2009

Dormid




Dormid may be available in the countries listed below.


Ingredient matches for Dormid



Midazolam

Midazolam is reported as an ingredient of Dormid in the following countries:


  • Argentina

International Drug Name Search

Sunday 5 July 2009

Cefuroxim-MIP




Cefuroxim-MIP may be available in the countries listed below.


Ingredient matches for Cefuroxim-MIP



Cefuroxime

Cefuroxime is reported as an ingredient of Cefuroxim-MIP in the following countries:


  • Poland

  • Serbia

Cefuroxime sodium salt (a derivative of Cefuroxime) is reported as an ingredient of Cefuroxim-MIP in the following countries:


  • Bulgaria

International Drug Name Search

After Bite




After Bite may be available in the countries listed below.


Ingredient matches for After Bite



Ammonium Hydroxide

Ammonium Hydroxide is reported as an ingredient of After Bite in the following countries:


  • Switzerland

International Drug Name Search